Pomares-Estran, Christelle, Delaunay, Pascal, Mottard, Annie, Cua, Eric, Roger, Pierre-Marie, Pradines, Bruno, ...
Abstract Endemic malaria has been eradicated from France, but some falciparum malaria cases have been described in patients who have never travelled outside the country. Ms. V. 21 year-old and Mr. M....
Malaria transmission in Dakar: A two-year survey (2008)
Pagès, Frederic, Texier, Gaetan, Pradines, Bruno, Gadiaga, Libasse, Machault, Vanessa, Jarjaval, Fanny, ...
Abstract Background According to entomological studies conducted over the past 30 years, there was low malaria transmission in suburb of Dakar but little evidence of it in the downtown area. However;...
Antimalarial drug use in general populations of tropical Africa (2008)
Gardella, Florence, Assi, Serge, Simon, Fabrice, Bogreau, Hervé, Eggelte, Teunis, Ba, Fatou, ...
Abstract Background The burden of Plasmodium falciparum malaria has worsened because of the emergence of chloroquine resistance. Antimalarial drug use and drug pressure are critical factors...
Briolant, Sébastien, Parola, Philippe, Fusaï, Thierry, Madamet-Torrentino, Marilyn, Baret, Eric, Mosnier, Joël, ...
Abstract Objective The main objective of this study was to assess the influence of gas mixtures on in vitro Plasmodium falciparum growth and 50% inhibitory concentration (IC 50 ) for chloroquine....
Daher, Wassim, Biot, Christophe, Fandeur, Thierry, Jouin, Helene, Pelinski, Lydie, Viscogliosi, Eric, ...
Abstract Background Ferroquine (FQ), or SSR97193, is a novel antimalarial drug currently in phase I clinical trials. FQ is a unique organometallic compound designed to overcome the chloroquine (CQ)...
Daher, Wassim, Biot, Christophe, Fandeur, Thierry, Jouin, Helene, Pelinski, Lydie, Viscogliosi, Eric, ...
BACKGROUND: Ferroquine (FQ), or SSR97193, is a novel antimalarial drug currently in phase I clinical trials. FQ is a unique organometallic compound designed to overcome the chloroquine (CQ)...
Daher, Wassim, Biot, Christophe, Fandeur, Thierry, Jouin, Helene, Pelinski, Lydie, Viscogliosi, Eric, ...
BACKGROUND: Ferroquine (FQ), or SSR97193, is a novel antimalarial drug currently in phase I clinical trials. FQ is a unique organometallic compound designed to overcome the chloroquine (CQ)...
Daher, Wassim, Biot, Christophe, Fandeur, Thierry, Jouin, Helene, Pelinski, Lydie, Viscogliosi, Eric, ...
BACKGROUND: Ferroquine (FQ), or SSR97193, is a novel antimalarial drug currently in phase I clinical trials. FQ is a unique organometallic compound designed to overcome the chloroquine (CQ)...
Daher, Wassim, Biot, Christophe, Fandeur, Thierry, Jouin, Helene, Pelinski, Lydie, Viscogliosi, Eric, ...
BACKGROUND: Ferroquine (FQ), or SSR97193, is a novel antimalarial drug currently in phase I clinical trials. FQ is a unique organometallic compound designed to overcome the chloroquine (CQ)...
Musset, Lise, Pradines, Bruno, Parzy, Daniel, Durand, Rémy, Bigot, Patricia, Le Bras, Jacques
Objectives: We examined the atovaquone in vitro susceptibility and the cytochrome b (cytb) gene polymorphism of African Plasmodium falciparum isolates during the first years of...
Musset, Lise, Pradines, Bruno, Parzy, Daniel, Durand, Rémy, Bigot, Patricia, Le Bras, Jacques
Objectives: We examined the atovaquone in vitro susceptibility and the cytochrome b (cytb) gene polymorphism of African Plasmodium falciparum isolates during the first years of atovaquone/proguanil...
Pradines, Bruno, Tall, Adama, Fusai, Thierry, Spiegel, Andre, Hienne, Remi, Rogier, Christophe, ...
The 50% inhibitory concentration (IC50s) of benflumetol (range, 12.5 to 240 nM; mean, 55.1 nM) for 158 Senegalese isolates were evaluated. Ten isolates (6%) showed decreased susceptibility to...
In Vitro Activities of Antibiotics against Plasmodium falciparum Are Inhibited by Iron
Pradines, Bruno, Rogier, Christophe, Fusai, Thierry, Mosnier, Joel, Daries, William, Barret, Eric, ...
The in vitro activities of cyclines (tetracycline, doxycycline, minocycline, oxytetracycline, and rolitetracycline), macrolides (erythromycin, spiramycin, roxithromycin, and lincomycin), quinolones...
Pradines, Bruno, Ramiandrasoa, Florence, Rolain, Jean Marc, Rogier, Christophe, Mosnier, Joel, Daries, William, ...
FR160, a catechol iron chelator, and tetracyclines or norfloxacin exert in vitro additive or synergistic activity against a chloroquine-resistant Plasmodium falciparum clone. FR160 shows antagonistic...
Pradines, Bruno, Alibert, Sandrine, Houdoin, Carole, Santelli-Rouvier, Christiane, Mosnier, Joel, Fusai, Thierry, ...
The effects of a series of dihydroethano- and ethenoanthracene derivatives on chloroquine (CQ) accumulation in CQ-susceptible strain 3D7 and CQ-resistant clone W2 were assessed. The levels of CQ...
Dihydroethanoanthracene Derivatives as In Vitro Malarial Chloroquine Resistance Reversal Agents
Millet, Julie, Torrentino-Madamet, Marylin, Alibert, Sandrine, Rogier, Christophe, Santelli-Rouvier, Christiane, Mosnier, Joel, ...
The ability of four 9,10-dihydroethanoanthracene derivatives (BG920, BG932, BG958, and BG996), as well as verapamil and promethazine, to reverse chloroquine resistance was assessed against 24...
Millet, Julie, Alibert, Sandrine, Torrentino-Madamet, Marylin, Rogier, Christophe, Santelli-Rouvier, Christiane, Bigot, Patricia, ...
BG958 reverses resistance in chloroquine-resistant isolates from different countries. Five mutations in the Plasmodium falciparum crt (pfcrt) gene resulting in the amino acid changes K76T, M74I,...
Daher, Wassim, Biot, Christophe, Fandeur, Thierry, Jouin, Helene, Pelinski, Lydie, Viscogliosi, Eric, ...
Pradines, Bruno, Hovette, Philippe, Fusai, Thierry, Atanda, Henri Léonard, Baret, Eric, Cheval, Philippe, ...
We determined the level of in vitro resistance of Plasmodium falciparum parasites to standard antimalarial drugs, such as chloroquine, quinine, amodiaquine, halofantrine, mefloquine, cycloguanil, and...
Pradines, Bruno, Tall, Adama, Fusai, Thierry, Spiegel, Andre, Hienne, Remi, Rogier, Christophe, ...
The 50% inhibitory concentration (IC50s) of benflumetol (range, 12.5 to 240 nM; mean, 55.1 nM) for 158 Senegalese isolates were evaluated. Ten isolates (6%) showed decreased susceptibility to...
In Vitro Activities of Antibiotics against Plasmodium falciparum Are Inhibited by Iron
Pradines, Bruno, Rogier, Christophe, Fusai, Thierry, Mosnier, Joel, Daries, William, Barret, Eric, ...
The in vitro activities of cyclines (tetracycline, doxycycline, minocycline, oxytetracycline, and rolitetracycline), macrolides (erythromycin, spiramycin, roxithromycin, and lincomycin), quinolones...
Pradines, Bruno, Ramiandrasoa, Florence, Rolain, Jean Marc, Rogier, Christophe, Mosnier, Joel, Daries, William, ...
FR160, a catechol iron chelator, and tetracyclines or norfloxacin exert in vitro additive or synergistic activity against a chloroquine-resistant Plasmodium falciparum clone. FR160 shows antagonistic...
Pradines, Bruno, Alibert, Sandrine, Houdoin, Carole, Santelli-Rouvier, Christiane, Mosnier, Joel, Fusai, Thierry, ...
The effects of a series of dihydroethano- and ethenoanthracene derivatives on chloroquine (CQ) accumulation in CQ-susceptible strain 3D7 and CQ-resistant clone W2 were assessed. The levels of CQ...
Dihydroethanoanthracene Derivatives as In Vitro Malarial Chloroquine Resistance Reversal Agents
Millet, Julie, Torrentino-Madamet, Marylin, Alibert, Sandrine, Rogier, Christophe, Santelli-Rouvier, Christiane, Mosnier, Joel, ...
The ability of four 9,10-dihydroethanoanthracene derivatives (BG920, BG932, BG958, and BG996), as well as verapamil and promethazine, to reverse chloroquine resistance was assessed against 24...
Millet, Julie, Alibert, Sandrine, Torrentino-Madamet, Marylin, Rogier, Christophe, Santelli-Rouvier, Christiane, Bigot, Patricia, ...
BG958 reverses resistance in chloroquine-resistant isolates from different countries. Five mutations in the Plasmodium falciparum crt (pfcrt) gene resulting in the amino acid changes K76T, M74I,...
Daher, Wassim, Biot, Christophe, Fandeur, Thierry, Jouin, Helene, Pelinski, Lydie, Viscogliosi, Eric, ...
Pradines, Bruno, Hovette, Philippe, Fusai, Thierry, Atanda, Henri Léonard, Baret, Eric, Cheval, Philippe, ...
We determined the level of in vitro resistance of Plasmodium falciparum parasites to standard antimalarial drugs, such as chloroquine, quinine, amodiaquine, halofantrine, mefloquine, cycloguanil, and...
Pradines, Bruno, Mamfoumbi, Modeste Mabika, Tall, Adama, Sokhna, Cheikh, Koeck, Jean-Louis, Fusai, Thierry, ...
Noranate, Nitchakarn, Durand, Rémy, Tall, Adama, Marrama, Laurence, Spiegel, André, Sokhna, Cheikh, ...
Briolant, Sébastien, Parola, Philippe, Fusaï, Thierry, Madamet-Torrentino, Marilyn, Baret, Eric, Mosnier, Joël, ...
Atorvastatin Is 10-Fold More Active In Vitro than Other Statins against Plasmodium falciparum▿
Pradines, Bruno, Torrentino-Madamet, Marylin, Fontaine, Albin, Henry, Maud, Baret, Eric, Mosnier, Joel, ...
Antimalarial drug use in general populations of tropical Africa
Gardella, Florence, Assi, Serge, Simon, Fabrice, Bogreau, Hervé, Eggelte, Teunis, Ba, Fatou, ...
Savini, Helene, Bogreau, Hervé, Bertaux, Lionel, Bouchiba, Housem, Kraemer, Philippe, Parzy, Daniel, ...
Malaria transmission in Dakar: A two-year survey
Pagès, Frederic, Texier, Gaetan, Pradines, Bruno, Gadiaga, Libasse, Machault, Vanessa, Jarjaval, Fanny, ...
Henry, Maud, Briolant, Sébastien, Fontaine, Albin, Mosnier, Joel, Baret, Eric, Amalvict, Rémy, ...
The in vitro activity of ferroquine (FQ) (SR97193), a 4-aminoquinoline antimalarial compound that contains a ferrocenic nucleus, against 15 Plasmodium falciparum strains was assessed and compared...
Briolant, Sébastien, Baragatti, Meili, Parola, Philippe, Simon, Fabrice, Tall, Adama, Sokhna, Cheikh, ...
The distribution and range of 50% inhibitory concentrations (IC50s) of doxycycline were determined for 747 isolates obtained between 1997 and 2006 from patients living in Senegal, Republic of the...
Pomares-Estran, Christelle, Delaunay, Pascal, Mottard, Annie, Cua, Eric, Roger, Pierre-Marie, Pradines, Bruno, ...
Endemic malaria has been eradicated from France, but some falciparum malaria cases have been described in patients who have never travelled outside the country. Ms. V. 21 year-old and Mr. M. 23...
Henry, Maud, Briolant, Sébastien, Zettor, Agnès, Pelleau, Stéphane, Baragatti, Meili, Baret, Eric, ...
Polymorphisms in the Plasmodium falciparum crt (Pfcrt), Pfmdr1, and Pfmrp genes were not significantly associated with quinine (QN) 50% inhibitory concentrations (IC50s) in 23 strains of Plasmodium...