James A. Lynham

Publication List Details

Period

2003 - 2003

Number

7

Co-Authors

(-)-CGP 12177 increases contractile force and hastens relaxation of human myocardial preparations through a propranolol-resistant state of the beta1-adrenoceptor (2003)

Sarsero, Doreen, Russell, Fraser D., Lynham, James A., Rabnott, Glenn, Yang, Ian, Fong, Kwun M., ...

Two forms of the activated beta(1)-adrenoceptor exist, one that is stabilized by (-)-noradrenaline and is sensitive to blockade by (-)-propranolol and another which is stabilized by partial agonists...

(-)-CGP 12177 increases contractile force and hastens relaxation of human myocardial preparations through a propranolol-resistant state of the beta1-adrenoceptor (2003)

Sarsero, Doreen, Russell, Fraser D., Lynham, James A., Rabnott, Glenn, Yang, Ian, Fong, Kwun M., ...

Two forms of the activated beta(1)-adrenoceptor exist, one that is stabilized by (-)-noradrenaline and is sensitive to blockade by (-)-propranolol and another which is stabilized by partial agonists...

Effects of collagen, ionophore A23187 and prostaglandin E1 on the phosphorylation of specific proteins in blood platelets

Haslam, Richard J., Lynham, James A., Fox, Joan E. B.

Human platelets that had been preincubated with 5-hydroxy[3H]tryptamine and [32P]Pi were stirred with various agents; the secretion of 5-hydroxy[3H]tryptamine from platelet granules and the...

Effects of collagen, ionophore A23187 and prostaglandin E1 on the phosphorylation of specific proteins in blood platelets

Haslam, Richard J., Lynham, James A., Fox, Joan E. B.

Human platelets that had been preincubated with 5-hydroxy[3H]tryptamine and [32P]Pi were stirred with various agents; the secretion of 5-hydroxy[3H]tryptamine from platelet granules and the...

Stimulation of cyclic AMP-dependent protein kinase in rat atria by (–;)-CGP 12177 through an atypical β-adrenoceptor

Kaumann, Alberto J, Lynham, James A

Mammalian hearts possess an atypical β-adrenoceptor (non-β1, non-β2, non-β3) through which (–)-4-(3-t-butylamino-2-hydroxypropoxy)benzimidazol-2-one ((–)-CGP 12177) causes cardiostimulant...

Comparison of the affinity of β-blockers for two states of the β1-adrenoceptor in ferret ventricular myocardium

Lowe, Martin D, Lynham, James A, Grace, Andrew A, Kaumann, Alberto J

We compared the potency of 11 clinically available β-blockers as antagonists of the positive inotropic effects of (−)-isoprenaline and CGP12177 on ferret ventricular myocardium.(−)-CGP12177,...

Octimibate, a potent non-prostanoid inhibitor of platelet aggregation, acts via the prostacyclin receptor

Merritt, Janet E., Hallam, Trevor J., Brown, Anthony M., Boyfield, Isobel, Cooper, David G., Hickey, Deirdre M.B., ...

1 Octimibate, 8-[(1,4,5-triphenyl-1H-imidazol-2-yl)oxy]octanoic acid, is reported to have antihrombotic properties, This is in addition to its antihyperlipidaemic effects which are due to inhibition...