Ring-substituted 4-Hydroxy-1H-quinolin-2-ones: Preparation and Biological Activity (2009)
Josef Jampilek, Robert Musiol, Matus Pesko, Katarina Kralova, Marcela Vejsova, James Carroll, ...
In the study, a series of twelve ring-substituted 4-hydroxy-1H-quinolin-2-one derivatives were prepared. The procedures for synthesis of the compounds are presented. The compounds were analyzed using...
Coupling Reactions of α-Bromocarboxylate with Non-Aromatic N-Heterocycles (2009)
Katerina Brychtova, Barbora Slaba, Lukas Placek, Josef Jampilek, Ivan Raich, Jozef Csollei
The conditions for the C-N bond forming reaction (C-N coupling reaction) between α-bromocarboxylate and nitrogen-containing non-aromatic heterocyclic rings under heterogeneous copper(I) oxide...
Jan Dolezel, Petra Hirsova, Veronika Opletalova, Jiri Dohnal, Vejsova Marcela, Jiri Kunes, ...
Some [(5Z)-(5-arylalkylidene-4-oxo-2-thioxo-1,3-thiazolidin-3-yl)]acetic acids were prepared as potential antifungal compounds. The general synthetic approach to all synthesized compounds is...
Investigating Biological Activity Spectrum for Novel Styrylquinazoline Analogues (2009)
Josef Jampilek, Robert Musiol, Jacek Finster, Matus Pesko, James Carroll, Katarina Kralova, ...
In this study, series of ring-substituted 2-styrylquinazolin-4(3H)-one and 4-chloro-2-styrylquinazoline derivatives were prepared. The syntheses of the discussed compounds are presented. The...
Salicylanilide Acetates: Synthesis and Antibacterial Evaluation (2007)
Jarmila Vinsova, Ales Imramovsky, Vladimir Buchta, Martina Ceckova, Martin Dolezal, Frantisek Staud, ...
A new series of salicylanilide acetates was synthesized and evaluated for their in vitro antifungal and antituberculotic activity. Some of the evaluated compounds possessed comparable or better...
Salicylanilide Acetates: Synthesis and Antibacterial Evaluation (2007)
Jarmila Vinsova, Ales Imramovsky, Vladimir Buchta, Martina Ceckova, Martin Dolezal, Frantisek Staud, ...
A new series of salicylanilide acetates was synthesized and evaluated for their in vitro antifungal and antituberculotic activity. Some of the evaluated compounds possessed comparable or better...
Substituted Pyrazinecarboxamides: Synthesis and Biological Evaluation (2006)
Martin Dolezal, Lukas Palek, Jarmila Vinsova, Vladimir Buchta, Josef Jampilek, Katarina Kralova
Condensation of the corresponding chlorides of some substituted pyrazine-2-carboxylic acids (pyrazine-2-carboxylic acid, 6-chloropyrazine-2-carboxylic acid, 5-tert-butylpyrazine-2-carboxylic acid or...