Robert H. Tukey

Human CYP1A1GFP Expression in Transgenic Mice Serves as a Biomarker for Environmental Toxicant Exposure (2007)

Operaña, Theresa N., Nguyen, Nghia, Chen, Shujuan, Beaton, Deirdre, Tukey, Robert H.

The human CYP1A1 gene is regulated by the aryl hydrocarbon receptor (AhR), and induction of CYP1A1 is known to play an important role in xenobiotic metabolism. To examine the regulation of human...

Human CYP1A1GFP Expression in Transgenic Mice Serves as a Biomarker for Environmental Toxicant Exposure (2006)

Operaña, Theresa N., Nguyen, Nghia, Chen, Shujuan, Beaton, Deirdre, Tukey, Robert H.

The human CYP1A1 gene is regulated by the aryl hydrocarbon receptor (AhR) and induction of CYP1A1 is known to play an important role in xenobiotic metabolism. To examine the regulation of human...

The Role of Protein Kinase C in Regulation of TCDD-Mediated CYP1A1 Gene Expression (2005)

Machemer, Daniel E. W., Tukey, Robert H.

Cytochrome P450 1A1 (CYP1A1) is induced by halogenated and polycyclic aromatic hydrocarbons following activation of the aryl hydrocarbon receptor (AhR). Protein kinase C (PKC) has been implicated in...

The Role of Protein Kinase C in Regulation of TCDD-Mediated CYP1A1 Gene Expression (2005)

Machemer, Daniel E.W., Tukey, Robert H.

Cytochrome P450 1A1 (CYP1A1) is induced by halogenated and polycyclic aromatic hydrocarbons following activation of the Ah receptor. Protein kinase C (PKC) has been implicated in the regulation of...

Mol Pharmacol 67:1247–1256, 2005 Printed in U.S.A. Arsenite Inhibition of CYP1A1 Induction by 2,3,7,8- Tetrachlorodibenzo-p-dioxin Is Independent of Cell Cycle Arrest (2004)

Jessica A. Bonzo, Shujuan Chen, Alema Galijatovic, Robert H. Tukey

We show here that arsenite (As 3 � ) elicits multiple effects on gene control, such as the interruption of cell cycle control by initiating G 2/M arrest as well as inhibiting the aryl hydrocarbon...

The contribution of UDP-glucuronosyltransferase 1A9 on CYP1A2-mediated genotoxicity by aromatic and heterocyclic amines (2001)

Yueh, Mei-Fei, Nguyen, Nghia, Famourzadeh, Maryam, Strassburg, Christian P., Oda, Yoshimitsu, Guengerich, F.Peter, ...

The importance of environmental and dietary arylamines, and heterocyclic amines in the etiology of human cancer is of growing interest. These pre-carcinogens are known to undergo bioactivation by...

Glucuronidation of 2-hydroxyamino-1-methyl-6-phenylimidazo[4,5-b]pyridine by human microsomal UDP-glucuronosyltransferases: identification of specific UGT1A family isoforms involved (1999)

Nowell, Susan A., Massengill, Joyce S., Williams, Suzanne, Radominska-Pandya, Anna, Tephly, Thomas R., Cheng, Ziqiang, ...

2-Amino-1-methyl-6-phenylimidazo[4,5-b]pyridine is a heterocyclic aromatic amine found in cooked meats and dietary exposure to PhIP has been implicated in the etiology of colon cancer in...

Activation of procarcinogens by human cytochrome P450 enzymes expressed in Escherichia coli. Simplified bacterial systems for genotoxicity assays (1994)

Shimada, Tsutomu, Gillam, Elizabeth M.J., Sandhu, Punam, Guo, Zuyu, Tukey, Robert H., Guengerich, F.Peter

Bacterial assays were used to examine the activation of 14 known procarcinogens by cytochrome P450 (P450) enzymest†. Human P450s 1A1, 1A2 and 3A4 were expressed in Escherichia coil with slight...

Control of steroid, heme, and carcinogen metabolism by nuclear pregnane X receptor and constitutive androstane receptor

Xie, Wen, Yeuh, Mei-Fei, Radominska-Pandya, Anna, Saini, Simrat P. S., Negishi, Yoichi, Bottroff, Bobbie Sue, ...

Through a multiplex promoter spanning 218 kb, the phase II UDP-glucuronosyltransferase 1A (UGT1) gene encodes at least eight differently regulated mRNAs whose protein products function as the...

Control of steroid, heme, and carcinogen metabolism by nuclear pregnane X receptor and constitutive androstane receptor

Xie, Wen, Yeuh, Mei-Fei, Radominska-Pandya, Anna, Saini, Simrat P. S., Negishi, Yoichi, Bottroff, Bobbie Sue, ...

Through a multiplex promoter spanning 218 kb, the phase II UDP-glucuronosyltransferase 1A (UGT1) gene encodes at least eight differently regulated mRNAs whose protein products function as the...