Zuyu Guo

Metabolism of 4-(methylnitrosamino)-1-(3-pyridyl)-1-butanone (NNK) by human cytochrome P450 1A2 and its inhibition by phenethyl isothiocyanate (1996)

Smith, Theresa J., Guo, Zuyu, Guengerich, F.Peter, Yang, Chung S.

4-(Methylnitrosamino)-1-(3-pyridyl)-1-butanone (NNK) is a potent tobacco-specific nitrosamine in animals and has been suggested to play a role in human tobacco-related cancers. Our previous study...

Activation of procarcinogens by human cytochrome P450 enzymes expressed in Escherichia coli. Simplified bacterial systems for genotoxicity assays (1994)

Shimada, Tsutomu, Gillam, Elizabeth M.J., Sandhu, Punam, Guo, Zuyu, Tukey, Robert H., Guengerich, F.Peter

Bacterial assays were used to examine the activation of 14 known procarcinogens by cytochrome P450 (P450) enzymest†. Human P450s 1A1, 1A2 and 3A4 were expressed in Escherichia coil with slight...

Structure-activity relationships of arylalkyl isothiocyanates for the inhibition of 4-(methylnitrosamino)-1-(3-pyridyl)-1-butanone metabolism and the modulation of xenobiotic-metabolizing enzymes in rats and mice (1993)

Guo, Zuyu, Smith, Theresa J., Wang, Erjia, Eklind, Karin I., Chung, Fung-Lung, Yang, Chung S.

Many arylalkyl isothiocyanates are potent inhibitors of 4-(methylnitrosamino)-1-(3-pyridyl)-1-butanone (NNK)-induced lung tumorigenesis in rats and mice. In the mouse, 4-phenylbutyl isothiocyanate...

Effects of phenethyl isothiocyanate, a carcinogenesis inhibitor, on xenobiotic-metabolizing enzymes and nitrosamine metabolism in rats (1992)

Guo, Zuyu, Smith, Theresa J., Wang, Erjia, Sadrieh, Nakissa, Ma, Qiang, Thomas, Paul E, ...

Phenethyl isothiocyanate (PEITC), a constituent of cruciferous vegetables, has been shown to inhibit chemical carcinogenesis, possibly due to its ability to block the activation or to enhance the...

Kinetics and enzyme involvement in the metabolism of 4-(methylnitrosamino)-1-(3-pyridyl)-1-butanone (NNK) in microsomes of rat lung and nasal mucosa (1992)

Smith, Theresa J., Guo, Zuyu, Jun-Hong, Yan, Ning, Shu M., Thomas, Paul E., Yang, Chung S.

The rat lung and nasal cavity are two target organs for carcinogenesis by 4-(methylnitrosamino)-1-(3-pyridyl)-1-butanone (NNK). In order to characterize further the enzymes involved in the...

Matabolism of 4-(methylnitrosamino)-1-(3-pyridyl)-1-butanone (NNK) by cytochrome P450IIB1 in a reconstituted system (1991)

Guo, Zuyu, Smith, Theresa J., Ishizaki, Hiroyuki, Yang, Chung S.

Several previous studies have suggested that cytochrome P450IIB1 is involved in the bioactivation of the tobaccospecific carcinogen, 4-(methylnitrosamino)-1-(3-pyridy1)-1-butanone (NNK), in rat as...